Home Tools
Log in
Cart

Search Result

Search Results for " ccr1 antagonist 10 "

2

Compounds

Cat No. Product Name Synonyms Targets
T28072 MLN-3897 AVE9897,AVE 9897,CCR1 antagonist 10,AVE-9897 CCR
MLN-3897 (CCR1 antagonist 10) is an orally active antagonist of CCR1 with a Ki of 2.3 nM for 125I-MIP-1α binding to THP-1 cell membranes. MLN-3897 inhibits Akt signaling and MM cell survival and proliferation.
T41016 Vercirnon sodium GSK-1605786 sodium,CCX282-Bsodium,Traficet-ENsodium
Vercirnon (GSK1605786A) sodium is an orally bioavailable, selective, and potent CCR9 antagonist. It effectively inhibits CCR9-mediated calcium mobilization and chemotaxis in Molt-4 cells, exhibiting IC50 values of 5.4 nM...
TargetMol